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Chemodex
Tianeptine sodium salt
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Product Details | |
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Synonyms | 7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid S,S-dioxide sodium salt; S-1574; Stablon |
Product Type | Chemical |
Properties | |
Formula | C21H24ClN2O4S . Na |
MW | 435.9 . 23.0 |
CAS | 30123-17-2 |
Source/Host Chemicals | Synthetic |
Purity Chemicals | ≥98% (T) |
Appearance | White to pale yellow solid. |
Solubility | Soluble in DMSO (20mg/ml), DMF (30mg/ml), ethanol (10mg/ml) and water (10mg/ml). |
Identity | Determined by 1H-NMR. |
Declaration | Manufactured by Chemodex. |
Other Product Data |
Click here for Original Manufacturer Product Datasheet |
InChi Key | ZLBSUOGMZDXYKE-UHFFFAOYSA-M |
Smiles | ClC(C=C1)=CC2=C1C(NCCCCCCC([O-])=O)C(C=CC=C3)=C3N(C)S2(=O)=O.[Na+] |
Shipping and Handling | |
Shipping | AMBIENT |
Short Term Storage | +20°C |
Long Term Storage | +20°C |
Handling Advice |
Keep under inert gas. Very hygroscopic. |
Use/Stability | Stable for at least 2 years after receipt when stored at RT. |
Documents | |
MSDS | Inquire |
Product Specification Sheet | |
Datasheet |
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Tianeptine is an atypical antidepressant with diverse actions, most notably on the glutamatergic system. It is a selective facilitator of 5-HT (serotonin) uptake in vitro and in vivo. It attenuates glutamate release and modulates the function of the AMPA receptor. Tianeptine also acts as an agonist of the μ-opioid receptor (EC50s = 194 and 641nM for human and mouse receptors, respectively). Might have anti-inflammatory properties through modulation of TLR and NLRP3 inflammasome signaling pathways.
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